[a]
Institute of Pharmaceutical Chemistry, Goethe University Frankfurt
Frankfurt 60438
Germany
[b]
Structural Genomics Consortium, BMLS, Goethe University Frankfurt
Frankfurt 60438
Germany
susanne.mueller-knapp@
123456bmls.de
[c]
Structural Genomics Consortium, University of Toronto
Toronto
Ontario
M5G 1L7
Canada
Cheryl.Arrowsmith@
123456uhnresearch.ca
[d]
University of Toronto
Toronto
Ontario
M5G 1L7
Canada
[e]
Department of Data Science, The Institute of Cancer Research
London
SM2 5NG
UK
[f]
CRUK ICR/Imperial Convergence Science Centre
London
SM2 5NG
UK
[g]
Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research
London SM2 5NG
UK
[h]
Monash Institute of Pharmaceutical Sciences, Monash University
Parkville
Victoria 3052
Australia
[i]
School of Pharmaceutical Sciences, Nanjing Tech University
No. 30 South Puzhu Road
Nanjing 211816
People's Republic of China
[j]
Research and Development, Bayer AG, Pharmaceuticals
42103 Wuppertal
Germany
[k]
Centre for Medicines Discovery, University of Oxford
Old Road Campus Research Building, Roosevelt Drive
Oxford OX3 7DQ
UK
[l]
Merck KGaA
Darmstadt
Germany
[m]
Alzheimer's Research UK Oxford Drug Discovery Institute, Centre for Medicines Discovery,
University of Oxford
Oxford
OX3 7FZ
UK
[n]
Institut Recherches de Servier
125 Chemin de Ronde
78290 Croissy
France
[o]
Discovery Research, Boehringer Ingelheim
55216 Ingelheim am Rhein
Germany
[p]
Early Drug Discovery Unit (EDDU), Montreal Neurological Institute-Hospital, McGill
University
Montreal
QC
Canada
[q]
School of Life Sciences, Division of Biological Chemistry and Drug Discovery, University
of Dundee
James Black Centre
Dundee
UK
[r]
Structural Genomics Consortium, UNC Eshelman School of Pharmacy
Chapel Hill
NC
USA
[s]
Lineberger Comprehensive Cancer Center, Department of Medicine, School of Medicine,
University of North Carolina at Chapel Hill
Chapel Hill
NC
27599
USA
[t]
Structural Genomics Consortium, Department of Medicine, Karolinska University Hospital
and Karolinska Institutet
Stockholm
Sweden
[u]
Nuvisan Innovation Campus Berlin GmbH
Müllerstraße 178
13353
Berlin
Germany
[v]
Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology
and Medicinal Chemistry, Eshelman School of Pharmacy, University of North Carolina
at Chapel Hill
Chapel Hill
NC
27599
USA
[w]
Institute for Protein Innovation
Boston
MA
USA
[x]
National Center for Advancing Translational Sciences, National Institutes of Health
Rockville
Maryland 20850
USA
[y]
Medicinal Chemistry, Global R&D, Merck Healthcare KGaA
Frankfurter Straße 250
64293
Darmstadt
Germany
[z]
Takeda California
9625 Towne Centre Drive
San Diego
California 92121
USA
[aa]
Science for Life Laboratory, Department of Oncology-Pathology
Karolinska Institutet
Stockholm
Sweden
[ab]
Institute of Bioinformatics and Department of Biochemistry and Molecular Biology,
University of Georgia
Athens
GA
USA
[ac]
Genentech, Inc.
1 DNA Way
South San Francisco
California 94080
USA
[ad]
Department of Cancer Biology and Chemical Biology Program, Dana-Farber Cancer Institute
450 Brookline Ave
Boston
MA 02215
USA
[ae]
CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences
Vienna
Austria
[af]
European Molecular Biology Laboratory, European Bioinformatics Institute
Wellcome Genome Campus, Hinxton
Cambridgeshire CB10 1SD
UK
[ag]
Strategic Innovation, Global R&D, Merck Healthcare KGaA
Frankfurter Straße 250
64293
Darmstadt
Germany
[ah]
Kennedy Institute of Rheumatology, NDORMS, University of Oxford
UK
[ai]
Neuroscience Drug Discovery Unit, Research, Takeda Pharmaceutical Company Limited
Fujisawa
Kanagawa
Japan
[aj]
Chemical Biology Laboratory, Center for Cancer Research, National Cancer Institute,
National Institutes of Health
Frederick
MD
USA
[ak]
LMU Munich, Department of Pharmacy, Chair of Pharmaceutical and Medicinal Chemistry
81377 Munich
Germany
[al]
Discovery Network Group, Pfizer Medicine Design
Cambridge
MA 02139
USA
[am]
Drugs for Neglected Diseases initiative
15 Chemin Camille Vidart
Geneva 1202
Switzerland
[an]
AbbVie
North Chicago
Illinois
USA
[ao]
Global Research Externalization, Takeda California, Inc.
9625 Towne Center Drive
San Diego
CA 92121
USA
[ap]
Department of Pharmacology & Toxicology, University of Toronto
Toronto
Ontario M5S 1A8
Canada
[aq]
Research and Development, Bayer AG, Pharmaceuticals
13353 Berlin
Germany
[ar]
Structural & Protein Sciences, Discovery Sciences, Janssen Research & Development
1400 McKean Rd
Spring House
PA 19477
USA
[as]
Division of Rheumatology, Department of Medicine Solna, Karolinska University Hospital
and Karolinska Institutet
Stockholm
Sweden
[at]
Center for Physiology and Pharmacology, Medical University of Vienna
Vienna
Austria
[au]
School of Pharmacy, University College London
London
WC1N 1AX
UK
[av]
Diamond Light Source Ltd
Harwell Science and Innovation Campus
Didcot OX11 0QX
UK
[aw]
Department of Biochemistry, University of Johannesburg
Auckland Park 2006
South Africa
[ax]
Research Complex at Harwell
Harwell Science and Innovation Campus
Didcot OX11 0FA
UK
[ay]
Princess Margaret Cancer Centre
Toronto
Ontario
M5G 1L7
Canada